• 3078 Citations
  • 31 h-Index
19992020

Research output per year

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Research Output

2011

Solution-phase parallel synthesis and SAR of homopiperazinyl analogs as positive allosteric modulators of mGlu4

Cheung, Y. Y., Zamorano, R., Blobaum, A. L., Weaver, C. D., Conn, P. J., Lindsley, C. W., Niswender, C. M. & Hopkins, C. R., Mar 14 2011, In : ACS Combinatorial Science. 13, 2, p. 159-165 7 p.

Research output: Contribution to journalArticle

4 Scopus citations

Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu 4) antagonist: Unexpected 'molecular switch' from a closely related mGlu 4 positive allosteric modulator

Utley, T., Haddenham, D., Salovich, J. M., Zamorano, R., Vinson, P. N., Lindsley, C. W., Hopkins, C. R. & Niswender, C. M., Dec 1 2011, In : Bioorganic and Medicinal Chemistry Letters. 21, 23, p. 6955-6959 5 p.

Research output: Contribution to journalArticle

16 Scopus citations

The discovery and characterization of ML218: A novel, centrally active T-Type calcium channel inhibitor with robust effects in STN neurons and in a rodent model of Parkinson's disease

Xiang, Z., Thompson, A. D., Brogan, J. T., Schulte, M. L., Melancon, B. J., Mi, D., Lewis, L. M., Zou, B., Yang, L., Morrison, R., Santomango, T., Byers, F., Brewer, K., Aldrich, J. S., Yu, H., Dawson, E. S., Li, M., McManus, O., Jones, C. K., Daniels, J. S. & 5 others, Hopkins, C. R., Xie, X. S., Conn, P. J., Weaver, C. D. & Lindsley, C. W., Dec 21 2011, In : ACS Chemical Neuroscience. 2, 12, p. 730-742 13 p.

Research output: Contribution to journalArticle

49 Scopus citations
2012

ACS chemical neuroscience molecule spotlight on begacestat (GSI-953)

Hopkins, C. R., Jan 18 2012, In : ACS Chemical Neuroscience. 3, 1, p. 3-4 2 p.

Research output: Contribution to journalReview article

25 Scopus citations

ACS chemical neuroscience molecule spotlight on BMS-708163

Hopkins, C. R., Mar 21 2012, In : ACS Chemical Neuroscience. 3, 3, p. 149-150 2 p.

Research output: Contribution to journalReview article

5 Scopus citations

ACS chemical neuroscience molecule spotlight on potiga (Ezogabine)

Hopkins, C. R., Aug 15 2012, In : ACS Chemical Neuroscience. 3, 8, p. 632 1 p.

Research output: Contribution to journalReview article

4 Scopus citations

ACS chemical neuroscience molecule spotlight on suvorexant

Hopkins, C. R., Sep 19 2012, In : ACS Chemical Neuroscience. 3, 9, p. 647-648 2 p.

Research output: Contribution to journalReview article

10 Scopus citations

Allosteric modulation of seven transmembrane spanning receptors: Theory, practice, and opportunities for central nervous system drug discovery

Melancon, B. J., Hopkins, C. R., Wood, M. R., Emmitte, K. A., Niswender, C. M., Christopoulos, A., Conn, P. J. & Lindsley, C. W., Feb 23 2012, In : Journal of Medicinal Chemistry. 55, 4, p. 1445-1464 20 p.

Research output: Contribution to journalReview article

169 Scopus citations
15 Scopus citations

Discovery of N-(4-methoxy-7-methylbenzo[d]thiazol-2-yl)isonicatinamide, ML293, as a novel, selective and brain penetrant positive allosteric modulator of the muscarinic 4 (M4) receptor

Salovich, J. M., Vinson, P. N., Sheffler, D. J., Lamsal, A., Utley, T. J., Blobaum, A. L., Bridges, T. M., Le, U., Jones, C. K., Wood, M. R., Scott Daniels, J., Jeffrey Conn, P., Niswender, C. M., Lindsley, C. W. & Hopkins, C. R., Aug 1 2012, In : Bioorganic and Medicinal Chemistry Letters. 22, 15, p. 5084-5088 5 p.

Research output: Contribution to journalArticle

29 Scopus citations

DMH1, a highly selective small molecule BMP inhibitor promotes neurogenesis of hiPSCs: Comparison of PAX6 and SOX1 expression during neural induction

Neely, M. D., Litt, M. J., Tidball, A. M., Li, G. G., Aboud, A. A., Hopkins, C. R., Chamberlin, R., Hong, C. C., Ess, K. C. & Bowman, A. B., Jun 20 2012, In : ACS Chemical Neuroscience. 3, 6, p. 482-491 10 p.

Research output: Contribution to journalArticle

58 Scopus citations

DMH1, a novel BMP small molecule inhibitor, increases cardiomyocyte progenitors and promotes cardiac differentiation in mouse embryonic stem cells

Ao, A., Hao, J., Hopkins, C. R. & Hong, C. C., Jul 27 2012, In : PloS one. 7, 7, e41627.

Research output: Contribution to journalArticle

36 Scopus citations

Identification and characterization of a compound that protects cardiac tissue from human Ether-à-go-go-related gene (hERG)-related drug-induced arrhythmias

Potet, F., Lorinc, A. N., Chaigne, S., Hopkins, C. R., Venkataraman, R., Stepanovic, S. Z., Lewis, L. M., Days, E., Sidorov, V. Y., Engers, D. W., Zou, B., Afshartous, D., George, A. L., Campbell, C. M., Balser, J. R., Li, M., Baudenbacher, F. J., Lindsley, C. W., Weaver, C. D. & Kupershmidt, S., Nov 16 2012, In : Journal of Biological Chemistry. 287, 47, p. 39613-39625 13 p.

Research output: Contribution to journalArticle

11 Scopus citations

Identification of (R)-N-(4-(4-methoxyphenyl)thiazol-2-yl)-1- tosylpiperidine-2-carboxamide, ML277, as a novel, potent and selective K v7.1 (KCNQ1) potassium channel activator

Mattmann, M. E., Yu, H., Lin, Z., Xu, K., Huang, X., Long, S., Wu, M., McManus, O. B., Engers, D. W., Le, U. M., Li, M., Lindsley, C. W. & Hopkins, C. R., Sep 15 2012, In : Bioorganic and Medicinal Chemistry Letters. 22, 18, p. 5936-5941 6 p.

Research output: Contribution to journalArticle

28 Scopus citations

Iterative experimental and virtual high-throughput screening identifies metabotropic glutamate receptor subtype 4 positive allosteric modulators

Mueller, R., Dawson, E. S., Niswender, C. M., Butkiewicz, M., Hopkins, C. R., Weaver, C. D., Lindsley, C. W., Conn, P. J. & Meiler, J., Sep 2012, In : Journal of Molecular Modeling. 18, 9, p. 4437-4446 10 p.

Research output: Contribution to journalArticle

9 Scopus citations
27 Scopus citations

The metabotropic glutamate receptor 4-positive allosteric modulator VU0364770 produces efficacy alone and in combination with L-DOPA or an adenosine 2A antagonist in preclinical rodent models of Parkinson's disease

Jones, C. K., Bubser, M., Thompson, A. D., Dickerson, J. W., Turle-Lorenzo, N., Amalric, M., Blobaum, A. L., Bridges, T. M., Morrison, R. D., Jadhav, S., Engers, D. W., Italiano, K., Bode, J., Daniels, J. S., Lindsley, C. W., Hopkins, C. R., Conn, P. J. & Niswender, C. M., Feb 2012, In : Journal of Pharmacology and Experimental Therapeutics. 340, 2, p. 404-421 18 p.

Research output: Contribution to journalArticle

74 Scopus citations
2013

Discovery of a selective M4 positive allosteric modulator based on the 3-amino-thieno[2,3-b]pyridine-2-carboxamide scaffold: Development of ML253, a potent and brain penetrant compound that is active in a preclinical model of schizophrenia

Le, U., Melancon, B. J., Bridges, T. M., Vinson, P. N., Utley, T. J., Lamsal, A., Rodriguez, A. L., Venable, D., Sheffler, D. J., Jones, C. K., Blobaum, A. L., Wood, M. R., Daniels, J. S., Conn, P. J., Niswender, C. M., Lindsley, C. W. & Hopkins, C. R., Jan 1 2013, In : Bioorganic and Medicinal Chemistry Letters. 23, 1, p. 346-350 5 p.

Research output: Contribution to journalArticle

24 Scopus citations

Dynamic subunit stoichiometry confers a progressive continuum of pharmacological sensitivity by KCNQ potassium channels

Yu, H., Lin, Z., Mattmann, M. E., Zou, B., Terrenoire, C., Zhang, H., Wu, M., McManus, O. B., Kass, R. S., Lindsley, C. W., Hopkins, C. R. & Li, M., May 21 2013, In : Proceedings of the National Academy of Sciences of the United States of America. 110, 21, p. 8732-8737 6 p.

Research output: Contribution to journalArticle

39 Scopus citations

Eliciting Renal Failure in Mosquitoes with a Small-Molecule Inhibitor of Inward-Rectifying Potassium Channels

Raphemot, R., Rouhier, M. F., Hopkins, C. R., Gogliotti, R. D., Lovell, K. M., Hine, R. M., Ghosalkar, D., Longo, A., Beyenbach, K. W., Denton, J. S. & Piermarini, P. M., May 29 2013, In : PloS one. 8, 5, e64905.

Research output: Contribution to journalArticle

42 Scopus citations

Further exploration of M1 allosteric agonists: Subtle structural changes abolish M1 allosteric agonism and result in pan-mAChR orthosteric antagonism

Sheffler, D. J., Sevel, C., Le, U., Lovell, K. M., Tarr, J. C., Carrington, S. J. S., Cho, H. P., Digby, G. J., Niswender, C. M., Conn, P. J., Hopkins, C. R., Wood, M. R. & Lindsley, C. W., Jan 1 2013, In : Bioorganic and Medicinal Chemistry Letters. 23, 1, p. 223-227 5 p.

Research output: Contribution to journalArticle

10 Scopus citations

Inhibition of the TRPC5 ion channel protects the kidney filter

Schaldecker, T., Kim, S., Tarabanis, C., Tian, D., Hakroush, S., Castonguay, P., Ahn, W., Wallentin, H., Heid, H., Hopkins, C. R., Lindsley, C. W., Riccio, A., Buvall, L., Weins, A. & Greka, A., Dec 2 2013, In : Journal of Clinical Investigation. 123, 12, p. 5298-5309 12 p.

Research output: Contribution to journalArticle

96 Scopus citations

Is there a path forward for mGlu2 positive allosteric modulators for the treatment of schizophrenia?

Hopkins, C. R., Feb 20 2013, In : ACS Chemical Neuroscience. 4, 2, p. 211-213 3 p.

Research output: Contribution to journalArticle

27 Scopus citations

Reversible inhibitors of regulators of G-protein signaling identified in a high-throughput cell-based calcium signaling assay

Storaska, A. J., Mei, J. P., Wu, M., Li, M., Wade, S. M., Blazer, L. L., Sjögren, B., Hopkins, C. R., Lindsley, C. W., Lin, Z., Babcock, J. J., McManus, O. B. & Neubig, R. R., Dec 2013, In : Cellular Signalling. 25, 12, p. 2848-2855 8 p.

Research output: Contribution to journalArticle

17 Scopus citations
47 Scopus citations
2014

Chemical modulation of mutant mGlu1 receptors derived from deleterious GRM1 mutations found in schizophrenics

Cho, H. P., Garcia-Barrantes, P. M., Brogan, J. T., Hopkins, C. R., Niswender, C. M., Rodriguez, A. L., Venable, D. F., Morrison, R. D., Bubser, M., Daniels, J. S., Jones, C. K., Conn, P. J. & Lindsley, C. W., Oct 17 2014, In : ACS chemical biology. 9, 10, p. 2334-2346 13 p.

Research output: Contribution to journalArticle

30 Scopus citations

Discovery and characterization of a potent and selective inhibitor of Aedes aegypti inward rectifier potassium channels

Raphemot, R., Rouhier, M. F., Swale, D. R., Days, E., Weaver, C. D., Lovell, K. M., Konkel, L. C., Engers, D. W., Bollinger, S. F., Hopkins, C., Piermarini, P. M. & Denton, J. S., Nov 6 2014, In : PloS one. 9, 11, 110772.

Research output: Contribution to journalArticle

27 Scopus citations

Discovery and characterization of ML398, a potent and selective antagonist of the D4 receptor with in vivo activity

Berry, C. B., Bubser, M., Jones, C. K., Hayes, J. P., Wepy, J. A., Locuson, C. W., Daniels, J. S., Lindsley, C. W. & Hopkins, C. R., Sep 11 2014, In : ACS Medicinal Chemistry Letters. 5, 9, p. 1060-1064 5 p.

Research output: Contribution to journalArticle

9 Scopus citations

Identification of positive allosteric modulators VU0155094 (ML397) and VU0422288 (ML396) reveals new insights into the biology of metabotropic glutamate receptor 7

Jalan-Sakrikar, N., Field, J. R., Klar, R., Mattmann, M. E., Gregory, K. J., Zamorano, R., Engers, D. W., Bollinger, S. R., Weaver, C. D., Days, E. L., Lewis, L. M., Utley, T. J., Hurtado, M., Rigault, D., Acher, F., Walker, A. G., Melancon, B. J., Wood, M. R., Lindsley, C. W., Conn, P. J. & 3 others, Xiang, Z., Hopkins, C. R. & Niswender, C. M., Dec 17 2014, In : ACS Chemical Neuroscience. 5, 12, p. 1221-1237 17 p.

Research output: Contribution to journalArticle

35 Scopus citations

Specific activin receptor-like kinase 3 inhibitors enhance liver regeneration

Tsugawa, D., Oya, Y., Masuzaki, R., Ray, K., Engers, D. W., Dib, M., Do, N., Kuramitsu, K., Ho, K., Frist, A., Yu, P. B., Bloch, K. D., Lindsley, C. W., Hopkins, C. R., Hong, C. C. & Karp, S. J., Dec 1 2014, In : Journal of Pharmacology and Experimental Therapeutics. 351, 3, p. 549-558 10 p.

Research output: Contribution to journalArticle

18 Scopus citations
2015

Activation of metabotropic glutamate receptor 7 is required for induction of long-term potentiation at SCCA1 synapses in the hippocampus

Klar, R., Walker, A. G., Ghose, D., Grueter, B. A., Engers, D. W., Hopkins, C. R., Lindsley, C. W., Xiang, Z., Conn, P. J. & Niswender, C. M., May 13 2015, In : Journal of Neuroscience. 35, 19, p. 7600-7615 16 p.

Research output: Contribution to journalArticle

21 Scopus citations

Advancing biological understanding and therapeutics discovery with small-molecule probes

Schreiber, S. L., Kotz, J. D., Li, M., Aubé, J., Austin, C. P., Reed, J. C., Rosen, H., White, E. L., Sklar, L. A., Lindsley, C. W., Alexander, B. R., Bittker, J. A., Clemons, P. A., De Souza, A., Foley, M. A., Palmer, M., Shamji, A. F., Wawer, M. J., McManus, O., Wu, M. & 26 others, Zou, B., Yu, H., Golden, J. E., Schoenen, F. J., Simeonov, A., Jadhav, A., Jackson, M. R., Pinkerton, A. B., Chung, T. D. Y., Griffin, P. R., Cravatt, B. F., Hodder, P. S., Roush, W. R., Roberts, E., Chung, D. H., Jonsson, C. B., Noah, J. W., Severson, W. E., Ananthan, S., Edwards, B., Oprea, T. I., Conn, P. J., Hopkins, C. R., Wood, M. R., Stauffer, S. R. & Emmitte, K. A., 2015, In : Cell. 161, 6, p. 1252-1265 14 p.

Research output: Contribution to journalReview article

80 Scopus citations

Discovery and characterization of 2-(cyclopropanesulfonamido)-n-(2-ethoxyphenyl)benzamide, ML382: A potent and selective positive allosteric modulator of MrgX1

Wen, W., Wang, Y., Li, Z., Tseng, P. Y., McManus, O. B., Wu, M., Li, M., Lindsley, C. W., Dong, X. & Hopkins, C. R., Jan 2015, In : ChemMedChem. 10, 1, p. 57-61 5 p.

Research output: Contribution to journalArticle

2 Scopus citations

Identification and characterization of ml352: A novel, noncompetitive inhibitor of the presynaptic choline transporter

Ennis, E. A., Wright, J., Retzlaff, C. L., McManus, O. B., Lin, Z., Huang, X., Wu, M., Li, M., Daniels, J. S., Lindsley, C. W., Hopkins, C. R. & Blakely, R. D., Mar 18 2015, In : ACS Chemical Neuroscience. 6, 3, p. 417-427 11 p.

Research output: Contribution to journalArticle

13 Scopus citations

Inhibition of BMP signaling suppresses metastasis in mammary cancer

Owens, P., Pickup, M. W., Novitskiy, S. V., Giltnane, J. M., Gorska, A. E., Hopkins, C. R., Hong, C. C. & Moses, H. L., May 7 2015, In : Oncogene. 34, 19, p. 2437-2449 13 p.

Research output: Contribution to journalArticle

55 Scopus citations

Pharmacological stimulation of metabotropic glutamate receptor type 4 in a rat model of Parkinson's disease and l-DOPA-induced dyskinesia: Comparison between a positive allosteric modulator and an orthosteric agonist

Iderberg, H., Maslava, N., Thompson, A. D., Bubser, M., Niswender, C. M., Hopkins, C. R., Lindsley, C. W., Conn, P. J., Jones, C. K. & Cenci, M. A., Aug 2015, In : Neuropharmacology. 95, p. 121-129 9 p., 5768.

Research output: Contribution to journalArticle

25 Scopus citations

Synthesis and structure-activity relationships of a series of 4-methoxy-3-(piperidin-4-yl)oxy benzamides as novel inhibitors of the presynaptic choline transporter

Bollinger, S. R., Engers, D. W., Ennis, E. A., Wright, J., Locuson, C. W., Lindsley, C. W., Blakely, R. D. & Hopkins, C. R., Apr 15 2015, In : Bioorganic and Medicinal Chemistry Letters. 25, 8, p. 1757-1760 4 p.

Research output: Contribution to journalArticle

3 Scopus citations
2016

An insecticide resistance-breaking mosquitocide targeting inward rectifier potassium channels in vectors of Zika virus and malaria

Swale, D. R., Engers, D. W., Bollinger, S. R., Gross, A., Inocente, E. A., Days, E., Kanga, F., Johnson, R. M., Yang, L., Bloomquist, J. R., Hopkins, C. R., Piermarini, P. M. & Denton, J. S., Nov 16 2016, In : Scientific reports. 6, 36954.

Research output: Contribution to journalArticle

31 Scopus citations

Bone morphogenetic protein signaling promotes tumorigenesis in a murine model of high-grade glioma

Hover, L. D., Owens, P., Munden, A. L., Wang, J., Chambless, L. B., Hopkins, C. R., Hong, C. C., Moses, H. L. & Abel, T. W., Jul 1 2016, In : Neuro-Oncology. 18, 7, p. 928-938 11 p.

Research output: Contribution to journalArticle

14 Scopus citations

Development and Antiparkinsonian Activity of VU0418506, a Selective Positive Allosteric Modulator of Metabotropic Glutamate Receptor 4 Homomers without Activity at mGlu2/4 Heteromers

Niswender, C. M., Jones, C. K., Lin, X., Bubser, M., Thompson Gray, A., Blobaum, A. L., Engers, D. W., Rodriguez, A. L., Loch, M. T., Daniels, J. S., Lindsley, C. W., Hopkins, C. R., Javitch, J. A. & Conn, P. J., Sep 21 2016, In : ACS Chemical Neuroscience. 7, 9, p. 1201-1211 11 p.

Research output: Contribution to journalArticle

30 Scopus citations

Discovery, characterization and biological evaluation of a novel (R)-4,4-difluoropiperidine scaffold as dopamine receptor 4 (D4R) antagonists

Jeffries, D. E., Witt, J. O., McCollum, A. L., Temple, K. J., Hurtado, M. A., Harp, J. M., Blobaum, A. L., Lindsley, C. W. & Hopkins, C. R., 2016, In : Bioorganic and Medicinal Chemistry Letters. 26, 23, p. 5757-5764 8 p.

Research output: Contribution to journalArticle

2 Scopus citations

Discovery, Synthesis, and Preclinical Characterization of N-(3-Chloro-4-fluorophenyl)-1H-pyrazolo[4,3-b]pyridin-3-amine (VU0418506), a Novel Positive Allosteric Modulator of the Metabotropic Glutamate Receptor 4 (mGlu4)

Engers, D. W., Blobaum, A. L., Gogliotti, R. D., Cheung, Y. Y., Salovich, J. M., Garcia-Barrantes, P. M., Daniels, J. S., Morrison, R., Jones, C. K., Soars, M. G., Zhuo, X., Hurley, J., Macor, J. E., Bronson, J. J., Conn, P. J., Lindsley, C. W., Niswender, C. M. & Hopkins, C. R., Sep 21 2016, In : ACS Chemical Neuroscience. 7, 9, p. 1192-1200 9 p.

Research output: Contribution to journalArticle

24 Scopus citations

Discovery and characterization of a novel series of N-phenylsulfonyl-1H-pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu4)

Gogliotti, R. D., Blobaum, A. L., Morrison, R. M., Daniels, J. S., Salovich, J. M., Cheung, Y. Y., Rodriguez, A. L., Loch, M. T., Conn, P. J., Lindsley, C. W., Niswender, C. M. & Hopkins, C. R., Jul 1 2016, In : Bioorganic and Medicinal Chemistry Letters. 26, 13, p. 2984-2987 4 p.

Research output: Contribution to journalArticle

5 Scopus citations

Discovery and optimization of a novel series of highly CNS penetrant M4 PAMs based on a 5,6-dimethyl-4-(piperidin-1-yl)thieno[2,3-d]pyrimidine core

Wood, M. R., Noetzel, M. J., Engers, J. L., Bollinger, K. A., Melancon, B. J., Tarr, J. C., Han, C., West, M., Gregro, A. R., Lamsal, A., Chang, S., Ajmera, S., Smith, E., Chase, P., Hodder, P. S., Bubser, M., Jones, C. K., Hopkins, C. R., Emmitte, K. A., Niswender, C. M. & 5 others, Wood, M. W., Duggan, M. E., Conn, P. J., Bridges, T. M. & Lindsley, C. W., Jul 1 2016, In : Bioorganic and Medicinal Chemistry Letters. 26, 13, p. 3029-3033 5 p.

Research output: Contribution to journalArticle

17 Scopus citations

Discovery of 3-aminopicolinamides as metabotropic glutamate receptor subtype 4 (mGlu4) positive allosteric modulator warheads engendering CNS exposure and in vivo efficacy

Gogliotti, R. D., Engers, D. W., Garcia-Barrantes, P. M., Panarese, J. D., Gentry, P. R., Blobaum, A. L., Morrison, R. D., Daniels, J. S., Thompson, A. D., Jones, C. K., Conn, P. J., Niswender, C. M., Lindsley, C. W. & Hopkins, C. R., Jun 15 2016, In : Bioorganic and Medicinal Chemistry Letters. 26, 12, p. 2915-2919 5 p.

Research output: Contribution to journalArticle

1 Scopus citations

Inhibitors of the bone morphogenetic protein (BMP) signaling pathway: a patent review (2008-2015)

Hopkins, C. R., Oct 2 2016, In : Expert Opinion on Therapeutic Patents. 26, 10, p. 1115-1128 14 p.

Research output: Contribution to journalReview article

11 Scopus citations

ML418: The First Selective, Sub-Micromolar Pore Blocker of Kir7.1 Potassium Channels

Swale, D. R., Kurata, H., Kharade, S. V., Sheehan, J., Raphemot, R., Voigtritter, K. R., Figueroa, E. E., Meiler, J., Blobaum, A. L., Lindsley, C. W., Hopkins, C. R. & Denton, J. S., Jul 20 2016, In : ACS Chemical Neuroscience. 7, 7, p. 1013-1023 11 p.

Research output: Contribution to journalArticle

8 Scopus citations

Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate Receptors

Lindsley, C. W., Emmitte, K. A., Hopkins, C. R., Bridges, T. M., Gregory, K. J., Niswender, C. M. & Conn, P. J., Jun 8 2016, In : Chemical Reviews. 116, 11, p. 6707-6741 35 p.

Research output: Contribution to journalReview article

100 Scopus citations

Synthesis and characterization of a series of chiral alkoxymethyl morpholine analogs as dopamine receptor 4 (D4R) antagonists

Witt, J. O., McCollum, A. L., Hurtado, M. A., Huseman, E. D., Jeffries, D. E., Temple, K. J., Plumley, H. C., Blobaum, A. L., Lindsley, C. W. & Hopkins, C. R., May 1 2016, In : Bioorganic and Medicinal Chemistry Letters. 26, 10, p. 2481-2488 8 p.

Research output: Contribution to journalArticle

10 Scopus citations

Validation of an improved scale for rating L-DOPA-induced dyskinesia in the mouse and effects of specific dopamine receptor antagonists

Sebastianutto, I., Maslava, N., Hopkins, C. R. & Cenci, M. A., Dec 1 2016, In : Neurobiology of Disease. 96, p. 156-170 15 p.

Research output: Contribution to journalArticle

21 Scopus citations