Allosteric modulation of seven transmembrane spanning receptors: Theory, practice, and opportunities for central nervous system drug discovery

Bruce J. Melancon, Corey R. Hopkins, Michael R. Wood, Kyle A. Emmitte, Colleen M. Niswender, Arthur Christopoulos, P. Jeffrey Conn, Craig W. Lindsley

Research output: Contribution to journalReview articlepeer-review

210 Scopus citations
Original languageEnglish (US)
Pages (from-to)1445-1464
Number of pages20
JournalJournal of Medicinal Chemistry
Volume55
Issue number4
DOIs
StatePublished - Feb 23 2012
Externally publishedYes

ASJC Scopus subject areas

  • Molecular Medicine
  • Drug Discovery

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